Patent details 
	
	
	
		
		
			EP1357928
		 
		
			
				Title:
				
					A NOVEL PHARMACEUTICAL COMPOUND AND METHODS OF MAKING AND USING SAME
				 
			
			
		
	
	
		
		
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				Basic Information 
				
					Publication number: 
					EP1357928 
					
						WO Application Number: 
						US2001043117 
					
					Type: 
					
						
							European Patent Granted for NL 
						
						
						
						
						
					
					
					
					Status: 
					
						
							Deemed not to be granted 
						
						
						
						
					
					
					
						Publication Title: 
						Title When Made Available For Viewing: 
						Reason Lapsed: 
						 
				
					Application number: 
					EP01273387.9 
					
						WO Publication Number: 
						WO2003020200 
					
					
					
						EPO Publication Language: 
						English 
					
					
					
						SPC Number: 
						
							
						 
					
					
					First Applicant Residence Country: 
					United States of America (US) 
					
						Publications: 
						 
				
				
				
				
				
				
				Dates 
				
					Filing date: 
					16/11/2001 
					
					
					Grant date: 
					16/11/2011 
					
					
						EP Publication Date: 
						16/11/2011 
						WO Publication Date: 
						Claims Translations Received Date: 
						Claims Translation B1 Received Date: 
						Claims Translation B2 Received Date: 
						Claims Translation B3 Received Date: 
						Lapsed By Non Payment Annual Fee Date: 
					Renunciation Date: 
					NullificationDate: 
					Published: 
						Due To Cession Date: 
						 
				
					Registration date: 
					16/11/2011 
					
						EP B1 Publication Date: 
						16/11/2011 
						EP B2 Publication Date: 
						EP B3 Publication Date: 
						Description Translation B1 Received Date: 
						Description Translation B2 Received Date: 
						Description Translation B3 Received Date: 
						Expiration date: 
						
					
					15/11/2021 
					Lapsed By Expiration Date: 
					Revocation Date: 
						Invalidity Date: 
						16/11/2011 
					
					
					
						Response To Novelty Search Report Received: 
						Patent Granting Request: 
						Lapsed date: 
						 
				
				
				
					Applicant/holder  
					
						
						
							From: 
							16/11/2011 
						 
						
							  
							  
						 
						
							  
							
								Name: 
								Shire LLC 
							 
							
								Address: 
								9200 Brookfield Court, FLORENCE, KY 41042, United States of America (US) 
							 
						
						
					
				
				
				
				
				
				
				
				
				
					Inventor 
					
						
						
							Name: 
							PICARIELLO, Thomas 
						 
						
							Address: 
							BLACKSBURG, VA 24060, United States of America (US) 
						 
					
				
				
				
				
				
				
				
				
				
					Priority 
					
						
							1 
						
						
							Priority Patent Number: 
							248617 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							2 
						
						
							Priority Patent Number: 
							248618 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							3 
						
						
							Priority Patent Number: 
							248619 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							4 
						
						
							Priority Patent Number: 
							248620 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							5 
						
						
							Priority Patent Number: 
							248737 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							6 
						
						
							Priority Patent Number: 
							248738 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							7 
						
						
							Priority Patent Number: 
							248621 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							8 
						
						
							Priority Patent Number: 
							248622 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							9 
						
						
							Priority Patent Number: 
							248623 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							10 
						
						
							Priority Patent Number: 
							248734 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							11 
						
						
							Priority Patent Number: 
							248735 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							12 
						
						
							Priority Patent Number: 
							248736 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							13 
						
						
							Priority Patent Number: 
							248739 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							14 
						
						
							Priority Patent Number: 
							248740 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							15 
						
						
							Priority Patent Number: 
							248741 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							16 
						
						
							Priority Patent Number: 
							248742 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							17 
						
						
							Priority Patent Number: 
							248750 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							18 
						
						
							Priority Patent Number: 
							248751 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							19 
						
						
							Priority Patent Number: 
							248752 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							20 
						
						
							Priority Patent Number: 
							248755 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							21 
						
						
							Priority Patent Number: 
							248758 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							22 
						
						
							Priority Patent Number: 
							248760 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							23 
						
						
							Priority Patent Number: 
							248762 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							24 
						
						
							Priority Patent Number: 
							248624 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							25 
						
						
							Priority Patent Number: 
							248626 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							26 
						
						
							Priority Patent Number: 
							248628 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							27 
						
						
							Priority Patent Number: 
							248633 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							28 
						
						
							Priority Patent Number: 
							248635 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							29 
						
						
							Priority Patent Number: 
							248638 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							30 
						
						
							Priority Patent Number: 
							248639 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							31 
						
						
							Priority Patent Number: 
							248641 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							32 
						
						
							Priority Patent Number: 
							248644 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							33 
						
						
							Priority Patent Number: 
							248646 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							34 
						
						
							Priority Patent Number: 
							248649 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							35 
						
						
							Priority Patent Number: 
							248652 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							36 
						
						
							Priority Patent Number: 
							248655 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							37 
						
						
							Priority Patent Number: 
							248657 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							38 
						
						
							Priority Patent Number: 
							248661 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							39 
						
						
							Priority Patent Number: 
							248610 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							40 
						
						
							Priority Patent Number: 
							248605 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							41 
						
						
							Priority Patent Number: 
							248612 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							42 
						
						
							Priority Patent Number: 
							248613 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							43 
						
						
							Priority Patent Number: 
							248614 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							44 
						
						
							Priority Patent Number: 
							248615 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							45 
						
						
							Priority Patent Number: 
							248616 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							46 
						
						
							Priority Patent Number: 
							248749 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							47 
						
						
							Priority Patent Number: 
							248753 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							48 
						
						
							Priority Patent Number: 
							248754 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							49 
						
						
							Priority Patent Number: 
							248757 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							50 
						
						
							Priority Patent Number: 
							248759 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							51 
						
						
							Priority Patent Number: 
							248761 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							52 
						
						
							Priority Patent Number: 
							248763 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							53 
						
						
							Priority Patent Number: 
							248625 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							54 
						
						
							Priority Patent Number: 
							248627 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							55 
						
						
							Priority Patent Number: 
							248629 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							56 
						
						
							Priority Patent Number: 
							248630 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							57 
						
						
							Priority Patent Number: 
							248631 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							58 
						
						
							Priority Patent Number: 
							248632 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							59 
						
						
							Priority Patent Number: 
							248634 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							60 
						
						
							Priority Patent Number: 
							248636 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							61 
						
						
							Priority Patent Number: 
							248637 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							62 
						
						
							Priority Patent Number: 
							248640 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							63 
						
						
							Priority Patent Number: 
							248642 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							64 
						
						
							Priority Patent Number: 
							248643 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							65 
						
						
							Priority Patent Number: 
							248645 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							66 
						
						
							Priority Patent Number: 
							248647 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							67 
						
						
							Priority Patent Number: 
							248648 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							68 
						
						
							Priority Patent Number: 
							248650 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							69 
						
						
							Priority Patent Number: 
							248651 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							70 
						
						
							Priority Patent Number: 
							248653 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							71 
						
						
							Priority Patent Number: 
							248654 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							72 
						
						
							Priority Patent Number: 
							248656 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							73 
						
						
							Priority Patent Number: 
							248658 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							74 
						
						
							Priority Patent Number: 
							248659 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							75 
						
						
							Priority Patent Number: 
							248660 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							76 
						
						
							Priority Patent Number: 
							248662 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							77 
						
						
							Priority Patent Number: 
							248663 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							78 
						
						
							Priority Patent Number: 
							248794 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							79 
						
						
							Priority Patent Number: 
							248795 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							80 
						
						
							Priority Patent Number: 
							248797 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							81 
						
						
							Priority Patent Number: 
							248796 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							82 
						
						
							Priority Patent Number: 
							248769 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							83 
						
						
							Priority Patent Number: 
							248768 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							84 
						
						
							Priority Patent Number: 
							248770 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							85 
						
						
							Priority Patent Number: 
							248776 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							86 
						
						
							Priority Patent Number: 
							248777 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							87 
						
						
							Priority Patent Number: 
							248771 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							88 
						
						
							Priority Patent Number: 
							248772 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							89 
						
						
							Priority Patent Number: 
							248685 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							90 
						
						
							Priority Patent Number: 
							248779 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							91 
						
						
							Priority Patent Number: 
							248782 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							92 
						
						
							Priority Patent Number: 
							248764 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							93 
						
						
							Priority Patent Number: 
							248774 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							94 
						
						
							Priority Patent Number: 
							248787 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							95 
						
						
							Priority Patent Number: 
							248767 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							96 
						
						
							Priority Patent Number: 
							248778 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							97 
						
						
							Priority Patent Number: 
							248780 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							98 
						
						
							Priority Patent Number: 
							248781 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							99 
						
						
							Priority Patent Number: 
							248783 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							100 
						
						
							Priority Patent Number: 
							248833 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							101 
						
						
							Priority Patent Number: 
							248765 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							102 
						
						
							Priority Patent Number: 
							248766 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							103 
						
						
							Priority Patent Number: 
							248773 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							104 
						
						
							Priority Patent Number: 
							248775 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							105 
						
						
							Priority Patent Number: 
							248786 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							106 
						
						
							Priority Patent Number: 
							248785 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							107 
						
						
							Priority Patent Number: 
							248784 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							108 
						
						
							Priority Patent Number: 
							248672 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							109 
						
						
							Priority Patent Number: 
							248674 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							110 
						
						
							Priority Patent Number: 
							248673 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							111 
						
						
							Priority Patent Number: 
							248678 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							112 
						
						
							Priority Patent Number: 
							248677 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							113 
						
						
							Priority Patent Number: 
							248676 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							114 
						
						
							Priority Patent Number: 
							248675 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							115 
						
						
							Priority Patent Number: 
							248679 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							116 
						
						
							Priority Patent Number: 
							248671 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							117 
						
						
							Priority Patent Number: 
							248680 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							118 
						
						
							Priority Patent Number: 
							248681 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							119 
						
						
							Priority Patent Number: 
							248682 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							120 
						
						
							Priority Patent Number: 
							248683 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							121 
						
						
							Priority Patent Number: 
							248684 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							122 
						
						
							Priority Patent Number: 
							248791 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							123 
						
						
							Priority Patent Number: 
							248793 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							124 
						
						
							Priority Patent Number: 
							248664 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							125 
						
						
							Priority Patent Number: 
							248665 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							126 
						
						
							Priority Patent Number: 
							248666 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							127 
						
						
							Priority Patent Number: 
							248667 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							128 
						
						
							Priority Patent Number: 
							248668 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							129 
						
						
							Priority Patent Number: 
							248669 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							130 
						
						
							Priority Patent Number: 
							248790 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							131 
						
						
							Priority Patent Number: 
							248792 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							132 
						
						
							Priority Patent Number: 
							248848 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							133 
						
						
							Priority Patent Number: 
							248849 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							134 
						
						
							Priority Patent Number: 
							248850 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							135 
						
						
							Priority Patent Number: 
							248851 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							136 
						
						
							Priority Patent Number: 
							248852 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							137 
						
						
							Priority Patent Number: 
							248853 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							138 
						
						
							Priority Patent Number: 
							248854 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							139 
						
						
							Priority Patent Number: 
							248855 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							140 
						
						
							Priority Patent Number: 
							248856 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							141 
						
						
							Priority Patent Number: 
							248857 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							142 
						
						
							Priority Patent Number: 
							248858 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							143 
						
						
							Priority Patent Number: 
							248594 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							144 
						
						
							Priority Patent Number: 
							248595 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							145 
						
						
							Priority Patent Number: 
							248596 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							146 
						
						
							Priority Patent Number: 
							248597 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							147 
						
						
							Priority Patent Number: 
							248598 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							148 
						
						
							Priority Patent Number: 
							248602 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							149 
						
						
							Priority Patent Number: 
							248756 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							150 
						
						
							Priority Patent Number: 
							248743 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							151 
						
						
							Priority Patent Number: 
							248744 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							152 
						
						
							Priority Patent Number: 
							248748 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							153 
						
						
							Priority Patent Number: 
							248747 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							154 
						
						
							Priority Patent Number: 
							248746 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							155 
						
						
							Priority Patent Number: 
							248745 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							156 
						
						
							Priority Patent Number: 
							248599 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							157 
						
						
							Priority Patent Number: 
							248789 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							158 
						
						
							Priority Patent Number: 
							248670 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							159 
						
						
							Priority Patent Number: 
							248524 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							160 
						
						
							Priority Patent Number: 
							248525 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							161 
						
						
							Priority Patent Number: 
							248526 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							162 
						
						
							Priority Patent Number: 
							248527 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							163 
						
						
							Priority Patent Number: 
							248528 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							164 
						
						
							Priority Patent Number: 
							248529 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							165 
						
						
							Priority Patent Number: 
							248531 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							166 
						
						
							Priority Patent Number: 
							248532 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							167 
						
						
							Priority Patent Number: 
							248533 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							168 
						
						
							Priority Patent Number: 
							248537 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							169 
						
						
							Priority Patent Number: 
							248538 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							170 
						
						
							Priority Patent Number: 
							248539 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							171 
						
						
							Priority Patent Number: 
							248540 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							172 
						
						
							Priority Patent Number: 
							248721 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							173 
						
						
							Priority Patent Number: 
							248722 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							174 
						
						
							Priority Patent Number: 
							248723 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							175 
						
						
							Priority Patent Number: 
							248724 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							176 
						
						
							Priority Patent Number: 
							248725 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							177 
						
						
							Priority Patent Number: 
							248726 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							178 
						
						
							Priority Patent Number: 
							248699 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							179 
						
						
							Priority Patent Number: 
							248700 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							180 
						
						
							Priority Patent Number: 
							248727 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							181 
						
						
							Priority Patent Number: 
							248730 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							182 
						
						
							Priority Patent Number: 
							248530 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							183 
						
						
							Priority Patent Number: 
							248728 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							184 
						
						
							Priority Patent Number: 
							248729 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							185 
						
						
							Priority Patent Number: 
							248731 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							186 
						
						
							Priority Patent Number: 
							248732 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							187 
						
						
							Priority Patent Number: 
							248733 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							188 
						
						
							Priority Patent Number: 
							248535 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							189 
						
						
							Priority Patent Number: 
							248536 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							190 
						
						
							Priority Patent Number: 
							248713 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							191 
						
						
							Priority Patent Number: 
							248714 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							192 
						
						
							Priority Patent Number: 
							248715 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							193 
						
						
							Priority Patent Number: 
							248716 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							194 
						
						
							Priority Patent Number: 
							248717 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							195 
						
						
							Priority Patent Number: 
							248718 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							196 
						
						
							Priority Patent Number: 
							248719 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							197 
						
						
							Priority Patent Number: 
							248720 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							198 
						
						
							Priority Patent Number: 
							248686 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							199 
						
						
							Priority Patent Number: 
							248688 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							200 
						
						
							Priority Patent Number: 
							248689 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							201 
						
						
							Priority Patent Number: 
							248710 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							202 
						
						
							Priority Patent Number: 
							248691 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							203 
						
						
							Priority Patent Number: 
							248692 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							204 
						
						
							Priority Patent Number: 
							248693 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							205 
						
						
							Priority Patent Number: 
							248694 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							206 
						
						
							Priority Patent Number: 
							248695 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							207 
						
						
							Priority Patent Number: 
							248696 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							208 
						
						
							Priority Patent Number: 
							248697 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							209 
						
						
							Priority Patent Number: 
							248698 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							210 
						
						
							Priority Patent Number: 
							248701 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							211 
						
						
							Priority Patent Number: 
							248702 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							212 
						
						
							Priority Patent Number: 
							248703 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							213 
						
						
							Priority Patent Number: 
							248704 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							214 
						
						
							Priority Patent Number: 
							248706 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							215 
						
						
							Priority Patent Number: 
							248707 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							216 
						
						
							Priority Patent Number: 
							248708 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							217 
						
						
							Priority Patent Number: 
							248709 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							218 
						
						
							Priority Patent Number: 
							248711 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							219 
						
						
							Priority Patent Number: 
							248712 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							220 
						
						
							Priority Patent Number: 
							248600 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							221 
						
						
							Priority Patent Number: 
							248601 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							222 
						
						
							Priority Patent Number: 
							248603 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							223 
						
						
							Priority Patent Number: 
							248604 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							224 
						
						
							Priority Patent Number: 
							248606 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							225 
						
						
							Priority Patent Number: 
							248608 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							226 
						
						
							Priority Patent Number: 
							248609 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							227 
						
						
							Priority Patent Number: 
							248611 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							228 
						
						
							Priority Patent Number: 
							248607 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
						
							229 
						
						
							Priority Patent Number: 
							248705 P 
							Priority Date: 
							16/11/2000 
							
						 
						
							Priority Country: 
							United States of America (US) 
							
						 
					
				
				
				
				
				
					Classification 
					
						
							Main IPC Class: 
							
								
									A61K 47/48 ;
							 
						
						
					 
				
				
				
					Publication 
					
						Bulletin 
						
							
								1 
							
							
								Bulletin Heading: 
								VRV 
								Journal edition number: 
								2012/09 
							 
							
								Publication date: 
								29/02/2012 
								Description: 
								Lapse or annulment 
							 
						
							
								2 
							
							
								Bulletin Heading: 
								EP2 
								Journal edition number: 
								2011/47 
							 
							
								Publication date: 
								23/11/2011 
								Description: 
								European patents granted for the Netherlands 
							 
						
					
					
						European Patent Bulletin 
						
							
							
								Issue number: 
								201146 
							 
							
								Publication date: 
								16/11/2011 
								Description: 
								Grant (B1) 
							 
						
					
				
				
				
				
				
				
				
				
				
				
				
				
				
				
				
			 
			
			
				
					
					
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